Products for Research Use Only

NVS-CECR2-1

CAT: 0013-GTR19244066-01Size: 100 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19244066-01Size:100 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
NVS-CECR2-1, a non-BET family Bromodomain (BRD) inhibitor, is a potent and selective cat eye syndrome chromosome region, candidate 2 (CECR2) inhibitor. NVS-CECR2-1 binds to CECR2 BRD with high affinity (IC50=47 nM; KD=80 nM) . NVS-CECR2-1 exhibits cytotoxic activity and induces apoptosis against various cancer cells by targeting CECR2 as well as via CECR2-independent mechanism.
CAS Number
1992047-61-6
Field of Research
Epigenetics & Chromatin
Purity
>98% (HPLC)
Solubility
In Vitro: DMSO : 66.67 mg/mL (134.50 mM; Ultrasonic)
Smiles
O=S (=O) (C1=NC (=CC (=N1) C2=CC=C3C (C=CN3C4CC (NC (C) (C) C4) (C) C) =C2) NC5CC5) CCC
Molecular Formula
C27H37N5O2S
Molecular Weight
495.68
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.