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CYT-1010

CAT: 0013-GTR19206117-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19206117-01Size:25 mg
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Description
CYT-1010 is a potent and selective mu-opioid receptor agonist, demonstrating high functional bias with an EC50 of 0.0053 nM for inhibiting cAMP production versus 13.1 nM for β-arrestin recruitment. This profile makes it a valuable research tool for investigating biased agonism, G-protein signaling pathways, and pain-related in vitro and in vivo studies.
CAS Number
213769-33-6
Field of Research
Metabolism Research, Neuroscience, Pharmacology & Drug Discovery
Smiles
C (C=1C=2C (NC1) =CC=CC2) [C@H]3C (=O) N[C@@H] (CC4=CC=CC=C4) C (=O) NCCCC[C@@H] (NC ([C@H] (CC5=CC=C (O) C=C5) N) =O) C (=O) N3
Molecular Formula
C35H40N6O5
Molecular Weight
624.73
Storage Conditions
-20°C
Notes
For research use only.

Chemical Information

Cyt-1010
CAS Number213769-33-6
PubChem CID44129692
IUPAC Name(2S)-2-amino-N-[(3S,6S,9R)-3-benzyl-6-(1H-indol-3-ylmethyl)-2,5,8-trioxo-1,4,7-triazacyclotridec-9-yl]-3-(4-hydroxyphenyl)propanamide
Molecular FormulaC35H40N6O5
Molecular Weight624.7
XLogP3.3
Topological Polar Surface Area178
Hydrogen Bond Donor Count7
Hydrogen Bond Acceptor Count6
Rotatable Bond Count8
Heavy Atom Count46
Formal Charge0
Complexity1030
SMILES
C1CCNC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](C1)NC(=O)[C@H](CC2=CC=C(C=C2)O)N)CC3=CNC4=CC=CC=C43)CC5=CC=CC=C5
InChI
InChI=1S/C35H40N6O5/c36-27(18-23-13-15-25(42)16-14-23)32(43)39-29-12-6-7-17-37-33(44)30(19-22-8-2-1-3-9-22)40-35(46)31(41-34(29)45)20-24-21-38-28-11-5-4-10-26(24)28/h1-5,8-11,13-16,21,27,29-31,38,42H,6-7,12,17-20,36H2,(H,37,44)(H,39,43)(H,40,46)(H,41,45)/t27-,29+,30-,31-/m0/s1
InChIKey
CFVGCGXJRNVTFP-LYXINOJLSA-N
Chemical Structure
2D Structure
2D structure of Cyt-1010
CAS: 213769-33-6
CID: 44129692
Formula: C35H40N6O5
MW: 624.7
Interactive 3D Structure
Loading 3D structure...
View on PubChemRaw 3D data
Computed Properties
PropertyValue
Molecular Weight624.7
XLogP33.3
Hydrogen Bond Donor Count7
Hydrogen Bond Acceptor Count6
Rotatable Bond Count8
Exact Mass624.30601840
Monoisotopic Mass624.30601840
Topological Polar Surface Area178 Ų
Heavy Atom Count46
Formal Charge0
Complexity1030
Isotope Atom Count0
Defined Atom Stereocenter Count4
Undefined Atom Stereocenter Count0
Defined Bond Stereocenter Count0
Undefined Bond Stereocenter Count0
Covalently-Bonded Unit Count1
Compound Is CanonicalizedYes

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Alternative Products

CatalogName
MBS5752968CYT-1010
MBS3845778-01CYT-1010 hydrochloride
A19176-25CYT-1010 25mg
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A19176-100CYT-1010 100mg
A19176-50CYT-1010 50mg
A19176-10CYT-1010 10mg
A19176-5CYT-1010 5mg
A21348-5CYT-1010 hydrochloride 5mg
A21348-25CYT-1010 hydrochloride 25mg

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