Products for Research Use Only

GLL 398

CAT: 0013-GTR19183880-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19183880-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
GLL 398 is a potent and selective oral estrogen receptor degrader, demonstrating an IC50 of 1.14 nM. It effectively inhibits tumor growth in breast cancer xenograft models, supporting its use in both in vitro mechanistic studies and in vivo preclinical research for hormone receptor-positive cancers.
CAS Number
2077980-80-2
Field of Research
Metabolism Research
Smiles
CC/C (C1=CC=CC=C1) =C (C2=CC=C (B (O) O) C=C2) /C3=CC=C (C=C3) /C=C/C (O) =O
Molecular Formula
C25H23BO4
Molecular Weight
398.26
Storage Conditions
-20°C
Notes
For research use only.