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Olcegepant

CAT: 0013-GTR19177312-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19177312-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Olcegepant (BIBN-4096) is a potent and highly selective small-molecule antagonist of the human CGRP1 receptor, exhibiting sub-nanomolar affinity (Ki = 14.4 pM) . It is widely used in migraine research to investigate CGRP receptor function in both in vitro binding assays and in vivo animal models of neurogenic inflammation and vasodilation.
CAS Number
204697-65-4
Product Name Alternative
BIBN 4096, BIBN 4096BS, BIBN4096, BIBN-4096, Calcitonin gene-related peptide receptor, CGRP1, CGRPReceptor, CGRP Receptor, Olcegepant, inhibit, Inhibitor, hCGRP
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
96.08% (May vary between batches)
Solubility
DMSO:23.81 mg/mL (27.38 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (2.3 mM)
Smiles
O=C1N (CC=2C (N1) =CC=CC2) C3CCN (C (N[C@H] (CC4=CC (Br) =C (O) C (Br) =C4) C (N[C@H] (C (=O) N5CCN (CC5) C=6C=CN=CC6) CCCCN) =O) =O) CC3
Molecular Formula
C38H47Br2N9O5
Molecular Weight
869.65
Storage Conditions
-20°C
Notes
For research use only.

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018736-01Olcegepant
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MBS3605155-01Olcegepant (hydrochloride)
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A11512-5Olcegepant 5mg
A11512-2Olcegepant 2mg

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