LBP1

• Description :

  LBP1 is an orally active and low brain penetrant CB1 receptor agonist. LBP1 exhibits significant anti-allodynic and anti-hyperalgesic effects in rodent models of neuropathic pain[1].

• UNSPSC :

  12352005

• Target :

  Cannabinoid Receptor

• Type :

  Reference compound

• Related Pathways :

  GPCR/G Protein; Neuronal Signaling

• Field of Research :

  Neurological Disease

• Assay Protocol :

  https://www.medchemexpress.com/lbp1.html

• Smiles :

  O=C(N)CN1CCN(CC2=NC(C3=CN(CC4CCOCC4)C5=C3C=CC=C5Cl)=NO2)CC1

• Molecular Formula :

  C23H29ClN6O3

• Molecular Weight :

  472.97

• References & Citations :

  [1]Adam J M, et al. Low brain penetrant CB1 receptor agonists for the treatment of neuropathic pain[J]. Bioorganic & medicinal chemistry letters, 2012, 22 (8) : 2932-2937.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• CAS Number :

  [1050478-18-6]