Products for Research Use Only

Racecadotril

CAT: 0013-GTR19162434-01Size: 100 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19162434-01Size:100 mg
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Description
Racecadotril, also known as acetorphan, is an antidiarrheal drug which acts as a peripherally acting enkephalinase inhibitor. (In Vivo) :In mice, following i.v. administration, Racecadotril is rapidly metabolized to Thiorphan; thus, 30 min after the injection only Thiorphan is recovered from the kidney whereas the parent compound Racecadotril is not detected.In rats 92% of a single-dose (10 mg/kg) of radioactively labeled Racecadotril is eliminated within 24 h.Racecadotril is a neutral endopeptidase (NEP) inhibitor with known antidiarrheal activity in animals. Orally administered Racecadotril (100 mg/kg) shows efficacy in a rat model of castor oil-induced diarrhea.
CAS Number
81110-73-8
Product Name Alternative
Acetorphan
Field of Research
Pharmacology & Drug Discovery
Purity
>98% (HPLC)
Solubility
DMSO: 22mg/ml (57.07 mM) ; Water: <1mg/ml; Ethanol: 77mg/ml (199.75 mM)
Smiles
CC (=O) SCC (CC1=CC=CC=C1) C (=O) NCC (=O) OCC1=CC=CC=C1
Molecular Formula
C21H23NO4S
Molecular Weight
385.49
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
Benzyl (3- (acetylthio) -2-benzylpropanoyl) glycinate

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