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BRL54443

CAT: 0013-GTR19161413-01Size: 200 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19161413-01Size:200 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
BRL54443 is a potent, releative selective 5-HT1E/1F agonist with Ki of 2/1 nM, respectively; shows low affinity for other receptors 5-HT1A (63 nM), 5-HT1B (126 nM), 5-HT1D (63 nM), 5-HT2A (1259 nM), 5-HT2B (100 nM), 5-HT2C (316 nM), 5-HT6 (>10,000 nM), 5-HT7 (>10,000 nM), D2 (501 nM), D3 (631 nM), and α1B-adrenoceptors (1259 nM) ; selectively stimulates 5-HT1E receptors and potently inhibits forskolin-dependent cAMP production with IC50 of 14 nM in DG membranes; significantly reduces formalin-induced flinching in rats.
CAS Number
57477-39-1
Product Name Alternative
BRL 54443 | BRL-54443
Purity
>98% (HPLC)
Solubility
DMSO: ≥ 51 mg/mL
Smiles
CN1CCC (C2=CNC3=C2C=C (O) C=C3) CC1
Molecular Formula
C14H18N2O
Molecular Weight
230.3055
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
1H-Indol-5-ol, 3- (1-methyl-4-piperidinyl) -

Alternative Products

CatalogName
MBS3605096-01BRL54443

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