Products for Research Use Only

ERK5-IN-2

CAT: 0013-GTR19169652-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19169652-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
ERK5-IN-2 is a selective, orally bioavailable ERK5 inhibitor with sub-micromolar potency, exhibiting IC50 values of 0.82 μM against ERK5 and 3 μM for the ERK5-MEF2D complex. This tool compound is used in biochemical and cellular assays to investigate the role of ERK5 signaling in cancer, inflammation, and cardiovascular disease research.
CAS Number
1888305-96-1
Product Name Alternative
Inhibit, ERK, ERK5IN2, ERK-5-IN-2, ERK5-IN-2, ERK5, ERK5 IN 2, Extracellular signal regulated kinases, Inhibitor
Field of Research
Signal Transduction, Stem Cell & Developmental Biology
Purity
≥95% (May vary between batches)
Solubility
DMSO:10 mg/mL (25.76 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:1 mg/mL (2.58 mM)
Smiles
Fc1cccc (Br) c1C (=O) c1c[nH]c (c1) C (=O) Nc1cccnc1
Molecular Formula
C17H11BrFN3O2
Molecular Weight
388.19
Storage Conditions
-20°C
Notes
For research use only.