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Alobresib

CAT: 0013-GTR19157931-01Size: 200 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19157931-01Size:200 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Alobresib is an inhibitor of BET bromodomain, is an antineoplastic drug candidate.in vitro experiments demonstrated high sensitivity of USC cell lines to the exposure to GS-5829, GS-626510, and JQ1 with BET inhibitors causing a dose-dependent decrease in the phosphorylated levels of c-Myc and a dose-dependent increase in caspase activation (apoptosis) . In comparative in vivo experiments, GS-5829 and/or GS-626510 were found more effective than JQ1 at the concentrations/doses used in decreasing tumor growth in both USC-ARK1 and USC-ARK2 mouse xenograft models.
CAS Number
1637771-14-2
Product Name Alternative
Vorolanib, GS-5829
Purity
>98% (HPLC)
Solubility
In Vitro: DMSO : 83.33 mg/mL (190.47 mM)
Smiles
Cc1noc (C) c1-c1cc (c2nc ([nH]c2c1) C1CC1) C (O) (c1ccccn1) c1ccccn1
Molecular Formula
C26H23N5O2
Molecular Weight
437.5
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.

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