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A-3 hydrochloride

CAT: 0013-GTR19156986-01Size: 1 gDry Ice: NoHazardous: No
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CAT#:0013-GTR19156986-01Size:1 g
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
A-3 hydrochloride is a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases. A-3 hydrochloride also inhibits PKC and casein kinase I with Ki values of 47 μM and 80 μM, respectively. A-3 hydrochloride against PKA (Ki=4.3 μM), casein kinase II (Ki=5.1 μM) and myosin light chain kinase (MLCK) (Ki=7.4 μM) .A-3 hydrochloride inhibits MLC-kinase competitively with respect to ATP and that the Ki value is 7.4 μM, and it is also a competitive inhibitor of cAMP-dependent protein kinase, cGMP-dependent protein kinase, protein kinase C, casein kinase I, and casein kinase II, with respect to ATP, exhibits Ki values of 4.3 μM, 3.8 μM, 47 μM, 80 μM, and 5.1 μM, respectively.
CAS Number
78957-85-4
Purity
>98% (HPLC)
Solubility
DMSO:125 mg/mL (389.14 mM; Need ultrasonic)
Smiles
Cl.NCCNS (=O) (=O) c1cccc2c (Cl) cccc12
Molecular Formula
C12H14Cl2N2O2S
Molecular Weight
321.22
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.

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