Products for Research Use Only

Breceptin

CAT: 0013-GTR19150428-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19150428-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Breceptin (B 9870) serves as an antagonist and partial agonist for bradykinin B1/B2 receptors (B1/B2R) . In rabbit jugular vein contraction assays, it functions as an irreversible B2R antagonist, inhibiting bradykinin-induced vasoconstriction. B-9870 exhibits partial agonist characteristics in HEK 293 cells with high rabbit B2R expression, activating ERK1/2 phosphorylation, calcium mobilization, arachidonic acid release, and receptor internalization. Breceptin is applicable in research on breast cancer and non-small cell lung cancer inhibition.
Molecular Weight
2815.33
Notes
For research use only.

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