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DS08210767

CAT: 0804-HY-125879-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-125879-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
DS08210767 is a highly potent, orally bioavailable PTHR1 antagonist with IC50 of 90 nM[1].
CAS Number
2376334-75-5
UNSPSC
12352005
Target
PTHR
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease; Endocrinology
Assay Protocol
https://www.medchemexpress.com/ds08210767.html
Purity
99.40
Solubility
DMSO : 5 mg/mL (ultrasonic; warming; heat to 80°C)
Smiles
CC1(N=C(C2=CC=C(C=C2N(C1=O)C3=CC=C(C=C3)NCCNC4CCOCC4)C#N)C5CCCCC5)C
Molecular Formula
C31H39N5O2
Molecular Weight
513.67
References & Citations
[1]Arai Y, et al. Discovery of novel PTHR1 antagonists: Design, synthesis, and structure activity relationships. Bioorg Med Chem Lett. 2019 Sep 15;29 (18) :2613-2616.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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CatalogName
T11101-01DS08210767

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