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PITCOIN4

CAT: 0804-HY-156406-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-156406-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PITCOIN4 is a highly selective Class II Alpha PI3K-C2α inhibitor. PITCOIN4 shows nanomolar inhibition of PI3K-C2α and >100-fold selectivity in a general kinase panel[1].
UNSPSC
12352005
Target
PI3K
Type
Reference compound
Related Pathways
PI3K/Akt/mTOR
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/pitcoin4.html
Purity
99.97
Solubility
DMSO : 125 mg/mL (ultrasonic)
Smiles
CC(C)(NC(CC1=CSC(NC(CSC(N2CCC3=CC=CC=C3)=NC4=C(C2=O)N=CC=N4)=O)=N1)=O)C5=CC=CC=C5
Molecular Formula
C30H29N7O3S2
Molecular Weight
599.73
References & Citations
[1]Murat Kücükdisli, et al. Structural Basis for Highly Selective Class II Alpha Phosphoinositide-3-Kinase Inhibition. J Med Chem. 2023 Oct 26;66 (20) :14278-14302.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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