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EST64454

CAT: 0804-HY-131914Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-131914Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
EST64454 (compound 9k) is a selective, orally active sigma-1 receptor antagonist with Ki 22 nM. EST64454 can be used to study pain[1].
CAS Number
1351438-26-0
UNSPSC
12352005
Target
Sigma Receptor
Type
Reference compound
Related Pathways
Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Assay Protocol
https://www.medchemexpress.com/est64454.html
Smiles
CC(N1CCN(CCOCC2=NN(C3=CC=C(F)C(F)=C3)C=C2)CC1)=O
Molecular Formula
C18H22F2N4O2
Molecular Weight
364.39
References & Citations
[1]Yeste S, et al. Preliminary in Vitro Assessment of the Potential of EST64454, a Sigma-1 Receptor Antagonist, for Pharmacokinetic Drug-Drug Interactions. Biol Pharm Bull. 2020;43 (1) :68-76.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
Sigma 1 Receptor

Alternative Products

CatalogName
MBS5764993EST64454
BUP02801EST64454 hydrochloride
555898EST64454 HCl
MBS5813450EST64454 free base
T9306-01EST64454 Maleic acid salt

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