Grapiprant

• Target :

  Prostaglandin Receptor

• Related Pathways :

  GPCR/G Protein|||Immunology/Inflammation

• Purity :

  0.9984

• Bioactivity :

  Grapiprant (AAT-007) is a selective EP4 receptor antagonist. Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor (IC50: 35 nM, Ki: 24 nM) .

• Smiles :

  CCc1nc2c(C)nc(C)cc2n1-c1ccc(CCNC(=O)NS(=O)(=O)c2ccc(C)cc2)cc1

• Molecular Formula :

  C26H29N5O3S

• Molecular Weight :

  491.61

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  415903-37-6