TAK-683

• CAS Number :

  872719-49-8

• Target :

  Others|||Kisspeptin

• Related Pathways :

  Others|||GPCR/G Protein

• Bioactivity :

  TAK-683 is an effective full KISS1 receptor agonist (IC50=170 pM) . TAK-683 is a nonapeptide metastin analog, shows agonistic activities to KISS1R (EC50: 0.96 nM and 1.6 nM for human and rat, respectively) .

• Smiles :

  C([C@@H](NC([C@@H](CC1=CC=C(O)C=C1)NC(C)=O)=O)C(N[C@H](C(N[C@H](C(N[C@@H](CC2=CC=CC=C2)C(NNC(N[C@H](C(N[C@H](C(N[C@@H](CC=3C=4C(NC3)=CC=CC4)C(N)=O)=O)CCCNC(NC)=N)=O)CC(C)C)=O)=O)=O)[C@@H](C)O)=O)CC(N)=O)=O)C=5C=6C(NC5)=CC=CC6

• Molecular Formula :

  C64H83N17O13

• Molecular Weight :

  1298.45

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C