D[Cha4]-AVP

• Target:

  Vasopressin Receptor

• Related Pathways:

  GPCR/G Protein

• Bioactivity:

  Potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 receptors respectively) . Stimulates ACTH and corticosterone secretion and exhibits negligible vasopressor activity in vivo.

• Smiles:

  C (=O) (N1[C@H] (C (N[C@@H] (CCCNC (=N) N) C (NCC (N) =O) =O) =O) CCC1) [C@H]2NC (=O) [C@H] (CC (N) =O) NC (=O) [C@H] (CC3CCCCC3) NC (=O) [C@H] (CC4=CC=CC=C4) NC (=O) [C@H] (CC5=CC=C (O) C=C5) NC (=O) CCSSC2

• Molecular Formula:

  C50H71N13O11S2

• Molecular Weight:

  1094.31

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  500170-27-4