CH 275

CAT: 0931-MF-0040189-01Size: 1 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0040189-01Size:1 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
174688-78-9
Target
Somatostatin
Related Pathways
GPCR/G Protein
Bioactivity
Potent somatostatin receptor 1 (sst1) agonist; displays selectivity for sst1 (IC50 values are 30.9 nM, 345 nM, > 1 ?M, > 10 ?M and > 10?M for human sst1, sst3, sst4, sst2 and sst5 respectively) . Attenuates somatostatin release in the rat nucleus accumbens.
Smiles
C(C=1C=2C(NC1)=CC=CC2)[C@@H]3C(=O)N[C@@H](CC4=CC=C(CNC(C)C)C=C4)C(=O)N[C@@]([C@@H](C)O)(C(=O)N[C@@H](CC5=CC=CC=C5)C(=O)N[C@@]([C@@H](C)O)(C(=O)N[C@@H](CO)C(=O)N[C@H](C(O)=O)CSSC[C@H](N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC6=CC=CC=C6)C(=O)N[C@@H](CC7=CC=CC=C7)C(=O)N3)[H])[H]
Molecular Formula
C74H96N14O15S2
Molecular Weight
1485.8
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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