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GR231118

CAT: 0931-TP2022Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-TP2022Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
158859-98-4
Target
Neuropeptide Y Receptor
Related Pathways
Neuroscience, GPCR/G Protein
Bioactivity
Potent neuropeptide Y (NPY) Y1 receptor antagonist (pA2 = 10 and 10.5 at rY1 and hY1, receptors respectively) . Also a potent and selective NPY Y4 receptor agonist (pEC50 values are 6.0, 8.6 and 6.1 for rY2, hY4 and rY5 receptors respectively) . Suppresses food intake in rats in vivo. Also has affinity for neuropeptide FF (NPFF) receptors in vitro (Ki = 43-73 nM) .
Smiles
O=C1N2[C@](C(=O)N[C@H](C(N[C@@H](CC3=CC=C(O)C=C3)C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CC4=CC=C(O)C=C4)C(N)=O)=O)CCCNC(=N)N)=O)CC(C)C)=O)CCCNC(=N)N)=O)=O)CNC(=O)CC[C@H](NC([C@H]([C@H](CC)C)N)=O)C(=O)N5C(C(=O)N[C@H](C(N[C@@H](CC6=CC=C(O)C=C6)C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CC7=CC=C(O)C=C7)C(N)=O)=O)CCCNC(=N)N)=O)CC(C)C)=O)CCCNC(=N)N)=O)=O)CNC(=O)CC[C@@H]1NC([C@H]([C@H](CC)C)N)=O)(CCC5)[H])(CCC2)[H]
Molecular Formula
C110H170N34O24
Molecular Weight
2352.77
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Alternative Products

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HY-P1321GR231118
MBS5817815GR231118 TFA
HY-P1321AGR231118 (TFA)

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