PG-931

• Target :

  Melanocortin Receptor

• Related Pathways :

  GPCR/G Protein|||Neuroscience

• Bioactivity :

  Potent and selective melanocortin 4 (MC4) receptor agonist (IC50 values are 0.58 and 55 nM for human MC4 and MC3 receptors respectively) . Produces a rapid and dose dependent restoration of cardiovascular and respiratory function in hemorrhage-shocked rats.

• Smiles :

  C(C=1C=2C(NC1)=CC=CC2)[C@H]3C(=O)N[C@H](C(=O)N4[C@H](C(N[C@@H]([C@@H](C)C)C(N)=O)=O)CCC4)CCCCNC(=O)C[C@H](NC([C@H](CCCC)NC(C)=O)=O)C(=O)N5[C@](C(=O)N[C@H](CC6=CC=CC=C6)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N3)(CCC5)[H]

• Molecular Formula :

  C59H85N15O11

• Molecular Weight :

  1180.41

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  667430-81-1