RVD-Hp?

• Target :

  Cannabinoid Receptor

• Related Pathways :

  GPCR/G Protein

• Bioactivity :

  N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. Increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. Also high affinity CB2 positive allosteric modulator (Ki = 50 nM) .

• Smiles :

  C([C@@H](NC([C@@H](NC([C@H](CCCNC(=N)N)N)=O)C(C)C)=O)CC(O)=O)(=O)N1[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CC2=CC=CC=C2)C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CC3=CN=CN3)C(O)=O)=O)CO)=O)CC(C)C)=O)CC(C)C)=O)CCCCN)=O)=O)CC(N)=O)=O)C(C)C)=O)CCC1

• Molecular Formula :

  C65H105N19O17

• Molecular Weight :

  1424.66

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  1193362-76-3