Dynorphin A (1-10)

• Target:

  Opioid Receptor|||iGluR

• Related Pathways:

  GPCR/G Protein|||Membrane transporter/Ion channel|||Neuroscience|||Endocrinology/Hormones

• Bioactivity:

  Dynorphin A (1-10), an endogenous opioid neuropeptide, interacts with the ?-opioid receptor by binding to its extracellular loop 2 and inhibits NMDA-activated current, demonstrating an IC50 value of 42.0 ?M.

• Smiles:

  C([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CC1=CC=CC=C1)NC(CNC(CNC([C@H](CC2=CC=C(O)C=C2)N)=O)=O)=O)=O)CC(C)C)=O)CCCNC(=N)N)=O)CCCNC(=N)N)=O)[C@H](CC)C)=O)CCCNC(=N)N)(=O)N3[C@H](C(O)=O)CCC3

• Molecular Formula:

  C57H91N19O12

• Molecular Weight:

  1234.45

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  79994-24-4