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TAK-448

CAT: 0931-TP1094-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-TP1094-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1234319-68-6
Target
Kisspeptin
Related Pathways
GPCR/G Protein
Bioactivity
TAK-448 (MVT-602), a potent and full KISS1R agonist with an IC50 of 460 pM and an EC50 of 632 pM, has been studied in trials for the treatment of Prostate Cancer, Low Testosterone, Prostatic Neoplasms, and Hypogonadotropic Hypogonadism.
Smiles
C([C@H](NC([C@@H](NC([C@@H](NC(NNC([C@H](CC1=CC=CC=C1)NC([C@@H](NC([C@@H](NC(=O)[C@H]2N(C([C@@H](CC3=CC=C(O)C=C3)NC(C)=O)=O)C[C@H](O)C2)CC(N)=O)=O)[C@@H](C)O)=O)=O)=O)CC(C)C)=O)CCCNC(NC)=N)=O)C(N)=O)C=4C=5C(NC4)=CC=CC5
Molecular Formula
C58H80N16O14
Molecular Weight
1225.36
Shipping Conditions
Ice Packs
Storage Temperature
-20°C