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4,5-Dimethoxycanthin-6-one

CAT: 0931-TN3013-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-TN3013-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
18110-87-7
Target
PDE, Cytochromes P450, Antibacterial
Related Pathways
Microbiology/Virology, Metabolism
Purity
0.9893
Bioactivity
4,5-Dimethoxycanthin-6-one is an alkaloid isolated from Picrasma quassioides BENNET (Simaroubaceae) with antimicrobial activity against Staphylococcus aureus and its drug-resistant strains. It is a potent, non-competitive inhibitor of CYP1A2-mediated phenacetin O-deethylation (IC50: 1.7 μM, Ki: 2.6 μM) and a potent inhibitor of cyclic adenosine monophosphate (cAMP) phosphodiesterase. Additionally, it exhibits cytotoxicity to tumor cell lines U937 and HepG2.
Smiles
COc1c(OC)c(=O)n2c3ccccc3c3ccnc1c23
Molecular Formula
C16H12N2O3
Molecular Weight
280.28
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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