Products for Research Use Only

SETDB1-TTD-IN-1

CAT: 0931-T9742-01Size: 1 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T9742-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
2755823-12-0
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Purity
0.9996
Bioactivity
SETDB1-TTD-IN-1 is a potent and selective inhibitor of SET domain bifurcated protein 1 tandem tudor domain (SETDB1-TTD, Kd = 88 nM), and also an endogenous binder competitive inhibitor with a KD of 0.106±0.002 μM for TTD. It can be used to study the biological functions and disease associations of SETDB1-TTD.
Smiles
CN1C[C@@H](C[C@@H](C1)c1ccc(OCc2ccccc2)cc1)Nc1nc2cc[nH]c2c(=O)n1CC=C
Molecular Formula
C28H31N5O2
Molecular Weight
469.58
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Popular Products