PF-04802367

CAT: 0931-T9611-01Size: 1 mgDry Ice: NoHazardous: No

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CAT#:0931-T9611-01Size:1 mg

Selected

24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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CAS Number

1962178-27-3

Target

GSK-3

Related Pathways

Stem Cells, PI3K/Akt/mTOR signaling

Purity

0.9876

Bioactivity

PF-04802367 is a highly selective GSK-3 inhibitor with an IC50 of 2.1 nM based on a recombinant human GSK-3β enzyme assay and 1.1 nM based on ADP-Glo assay. It shows desirable central nervous system (CNS) properties and potency. It is equally effective at inhibition of the two known GSK-3 isoforms (GSK-3α and GSK-3β) with IC50 values of 10.0 and 9.0 nM in mobility shift assays, respectively.

Smiles

COc1ccc(cc1Cl)-c1ocnc1C(=O)NCCCn1cncn1

Molecular Formula

C16H16ClN5O3

Molecular Weight

361.78

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

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PF-04802367

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