Borussertib

CAT: 0931-T8427-01Size: 1 mgDry Ice: NoHazardous: No

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CAT#:0931-T8427-01Size:1 mg

Selected

24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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CAS Number

1800070-77-2

Target

Akt

Related Pathways

Cytoskeletal Signaling, PI3K/Akt/mTOR signaling

Purity

0.99

Bioactivity

Borussertib is a first-in-class covalent-allosteric inhibitor of protein kinase Akt, with an IC50 of 0.8 nM and a Ki of 2.2 nM for Aktwt.

Smiles

C=CC(=O)Nc1ccc2[nH]c(=O)n(C3CCN(Cc4ccc(cc4)-c4nc5cc[nH]c(=O)c5cc4-c4ccccc4)CC3)c2c1

Molecular Formula

C36H32N6O3

Molecular Weight

596.68

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Alternative Products