Gestrinone

• Target :

  Estrogen/progestogen Receptor|||Estrogen Receptor/ERR

• Related Pathways :

  Endocrinology/Hormones

• Purity :

  0.9921

• Bioactivity :

  Gestrinone (R 2323) is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis. It inhibits leiomyoma cells with an IC50 of 43.67 ?M.

• Smiles :

  [H][C@@]12CC[C@@](O)(C#C)[C@@]1(CC)C=CC1=C3CCC(=O)C=C3CC[C@@]21[H]

• Molecular Formula :

  C21H24O2

• Molecular Weight :

  308.41

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  16320-04-0