Gestrinone

• Target:

  Estrogen/progestogen Receptor|||Estrogen Receptor/ERR

• Related Pathways:

  Endocrinology/Hormones

• Purity:

  0.9921

• Bioactivity:

  Gestrinone (R 2323) is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis. It inhibits leiomyoma cells with an IC50 of 43.67 ?M.

• Smiles:

  [H][C@@]12CC[C@@](O)(C#C)[C@@]1(CC)C=CC1=C3CCC(=O)C=C3CC[C@@]21[H]

• Molecular Formula:

  C21H24O2

• Molecular Weight:

  308.41

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  16320-04-0