Products for Research Use Only

Gestrinone

CAT: 0931-T7223-01Size: 1 mL - 10 mM (in DMSO)Dry Ice: NoHazardous: No
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CAT#:0931-T7223-01Size:1 mL - 10 mM (in DMSO)
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
16320-04-0
Target
Estrogen/progestogen Receptor, Estrogen Receptor/ERR
Related Pathways
Endocrinology/Hormones
Purity
0.9921
Bioactivity
Gestrinone (R 2323) is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to treat endometriosis. It inhibits leiomyoma cells with an IC50 of 43.67 μM.
Smiles
[H][C@@]12CC[C@@](O)(C#C)[C@@]1(CC)C=CC1=C3CCC(=O)C=C3CC[C@@]21[H]
Molecular Formula
C21H24O2
Molecular Weight
308.41
Shipping Conditions
Ice Packs
Storage Temperature
-20°C