Teneligliptin hydrobromide
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


Teneligliptin hydrobromide
Target:
Interleukin|||ROS|||DPP-4|||NF-?B|||Proteasome|||p38 MAPK|||Apoptosis|||AMPK|||JNK|||NOD-like Receptor (NLR) |||Immunology/Inflammation relatedRelated Pathways:
Proteases/Proteasome|||Chromatin/Epigenetic|||NF-?B|||PI3K/Akt/mTOR signaling|||Immunology/Inflammation|||Ubiquitination|||MAPK|||ApoptosisPurity:
>99.99%Bioactivity:
Teneligliptin hydrobromide (MP-513 (hydrobromide) ) is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50 values of approximately 1 nM.Smiles:
Br.Br.Br.Br.Br.Cc1cc(N2CCN(CC2)C2CNC(C2)C(=O)N2CCSC2)n(n1)-c1ccccc1.Cc1cc(N2CCN(CC2)C2CNC(C2)C(=O)N2CCSC2)n(n1)-c1ccccc1Molecular Formula:
C22H30N6OS·5/2BrHMolecular Weight:
628.86Shipping Conditions:
Cool packStorage Temperature:
-20°CCAS Number:
906093-29-6
