RS-127445
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


RS-127445
Target:
5-HT ReceptorRelated Pathways:
Neuroscience|||GPCR/G ProteinPurity:
0.9932Bioactivity:
RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.Smiles:
CC (C) c1cc (nc (N) n1) -c1ccc (F) c2ccccc12Molecular Formula:
C17H16FN3Molecular Weight:
281.33Shipping Conditions:
Cool packStorage Temperature:
-20°CCAS Number:
199864-87-4
