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GRPR antagonist-1

CAT: 0931-T63947-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T63947-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Others, Bombesin Receptor
Related Pathways
GPCR/G Protein, Others
Bioactivity
GRPR antagonist-1 is a potent antagonist of the gastrin-releasing peptide receptor (GRPR) and displays cytotoxicity to certain cancer cells, including PC3 cells (IC50: 4.97 μM), Pan02 cells (IC50: 4.36 μM), and HGC-27 cells (IC50: 3.40 μM) . It reduces Bcl-2 levels, increases Bax levels, inhibits HGC-27 cell viability, and induces apoptosis, thereby exhibiting anti-cancer effects.
Molecular Formula
C29H33F3N4O4
Molecular Weight
558.59
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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Alternative Products

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HY-115975GRPR antagonist-2
sc-398549GRPR (D-1)
sc-398549 FITCGRPR (D-1) FITC
sc-398549 ACGRPR (D-1) AC
sc-398549 HRPGRPR (D-1) HRP
HY-168633PSMA/GRPR ligand 1
sc-398549 PEGRPR (D-1) PE
sc-398549 AF680GRPR (D-1) Alexa Fluor® 680

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