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TGR5 Receptor Agonist 3

CAT: 0931-T63554-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T63554-01Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2643391-08-4
Target
Others, GPCR19
Related Pathways
GPCR/G Protein, Others
Bioactivity
TGR5 Receptor Agonist 3 is a G protein-coupled bile acid receptor 1 (GPBAR1, TGR5) agonist soft drug compound that decreases gallbladder filling, exhibits good gallbladder safety, and is able to act on hTGR5 (EC50: 16.4 nM) and mTGR5 (EC50: 209 nM) .
Smiles
C(=O)(N1C=2C(N(CC1)C3CC3)=CC=CC2)C=4C(OC=5C=C6C(=CC5)OC=C6C(OCOCC)=O)=CC=NC4
Molecular Formula
C29H27N3O6
Molecular Weight
513.54
Shipping Conditions
Ice Packs
Storage Temperature
-20°C