Y08284

• Target :

  Epigenetic Reader Domain|||Others

• Related Pathways :

  Others|||Chromatin/Epigenetic

• Bioactivity :

  Y08284 is a selective, potent, orally active inhibitor of CBP bromodomain (IC50: 4.21 nM) that inhibits the proliferation of prostate cancer cell lines LNCaP, C4-2B, and 22Rv1 and has anti-tumour effects.

• Smiles :

  C(NC1=C(F)C(=CC(C(C)O)=C1)C2=CN(N=C2)C3CC3)(=O)C4=C5N(C(C(C)=O)=C4)C=CC(OC)=C5

• Molecular Formula :

  C26H25FN4O4

• Molecular Weight :

  476.5

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  2688745-47-1