UNC9994 hydrochloride

CAT: 0931-MF-0039870-01Size: 2 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0039870-01Size:2 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2108826-33-9
Target
5-HT Receptor|||Dopamine Receptor|||Arrestin|||Others
Related Pathways
Neuroscience|||GPCR/G Protein|||Others
Bioactivity
UNC9994 hydrochloride is a functionally selective, ?-arrestin-biased dopamine D2 receptor (D2R) agonist (Ki: 79 nM) that selectively activates ?-arrestin recruitment and signal transduction. UNC9994 hydrochloride is a Gi-regulated antagonist of cAMP production and a partial agonist of the D2R/?-arrestin-2 interaction, exhibiting psychostimulatory effects.
Smiles
Cl.Clc1cccc(C2CCN(CCCOc3ccc4scnc4c3)CC2)c1Cl
Molecular Formula
C21H23Cl3N2OS
Molecular Weight
457.84
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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