Products for Research Use Only

Cabotegravir sodium

CAT: 0931-T62328-01Size: 1 mL - 10 mM (in DMSO)Dry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T62328-01Size:1 mL - 10 mM (in DMSO)
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
1051375-13-3
Target
Others, HIV Protease, OAT
Related Pathways
Membrane transporter/Ion channel, Others, Microbiology/Virology, Proteases/Proteasome
Purity
0.9963
Bioactivity
Cabotegravir sodium (GSK-1265744) is an orally active, membrane-permeable HIV integrase inhibitor (IC50 = 2.5 μM) and also an OAT1/OAT3 inhibitor (IC50 = 0.81/0.41 μM) . It inhibits HIV replication and may be used in AIDS research.
Smiles
[Na+].C[C@H]1CO[C@@H]2Cn3cc(C(=O)NCc4ccc(F)cc4F)c(=O)c([O-])c3C(=O)N12
Molecular Formula
C19H16F2N3NaO5
Molecular Weight
427.34
Shipping Conditions
Ice Packs
Storage Temperature
-20°C