LP-922761 hydrate

• Target:

  Others|||AAK1 (AP2 associated kinase 1)

• Related Pathways:

  Others|||Neuroscience

• Bioactivity:

  LP-922761 hydrate is a selective, potent, orally active AAK1 inhibitor with IC50 values of 4.8 nM and 7.6 nM in enzyme and cellular assays, respectively. LP-922761 hydrate inhibits BMP-2 inducible protein kinase (BIKE) (IC50: 24 nM) . 922761 hydrate has no significant effect on cellular GAK, opioids, adrenergic ?2 or GABAa receptors.

• Molecular Formula:

  C21H28N6O4

• Molecular Weight:

  414.98

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C