Darapladib

• Target:

  Phospholipase|||Apoptosis

• Related Pathways:

  Apoptosis|||Metabolism

• Purity:

  >99.99%

• Bioactivity:

  Darapladib (SB-480848) is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with an IC50 value of 0.25 nM, which can exert cardiovascular protective effects [1,3].

• Smiles:

  C(C(N(CC1=CC=C(C=C1)C2=CC=C(C(F)(F)F)C=C2)CCN(CC)CC)=O)N3C4=C(C(=O)N=C3SCC5=CC=C(F)C=C5)CCC4

• Molecular Formula:

  C36H38F4N4O2S

• Molecular Weight:

  666.77

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  356057-34-6