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Pilsicainide

CAT: 0931-T60482-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T60482-01Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
88069-67-4
Target
Sodium Channel, Others
Related Pathways
Others, Membrane transporter/Ion channel
Bioactivity
Pilsicainide (SUN 1165 free acid) is a potent class Ic antiarrhythmic agent and a sodium channel blocker[1][2].
Smiles
C(C(NC1=C(C)C=CC=C1C)=O)C23N(CCC2)CCC3
Molecular Formula
C17H24N2O
Molecular Weight
272.39
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

Chemical Information

Pilsicainide

Pilsicainide is a secondary carboxamide resulting from the formal condensation of the amino group of 2,6-dimethylaniline with the carboxy group of (tetrahydro-1H-pyrrolizin-7a(5H)-yl)acetic acid. It is a sodium channel blocker which is used as an antiarrhythmic drug for the management of atrial tachyarrhythmias in Japan. It has a role as an anti-arrhythmia drug and a sodium channel blocker. It is a secondary carboxamide and an organic heterobicyclic compound.

CAS Number88069-67-4
PubChem CID4820
IUPAC NameN-(2,6-dimethylphenyl)-2-(1,2,3,5,6,7-hexahydropyrrolizin-8-yl)acetamide
Molecular FormulaC17H24N2O
Molecular Weight272.4
XLogP2.7
Topological Polar Surface Area32.3
Hydrogen Bond Donor Count1
Hydrogen Bond Acceptor Count2
Rotatable Bond Count3
Heavy Atom Count20
Formal Charge0
Complexity348
SMILES
CC1=C(C(=CC=C1)C)NC(=O)CC23CCCN2CCC3
InChI
InChI=1S/C17H24N2O/c1-13-6-3-7-14(2)16(13)18-15(20)12-17-8-4-10-19(17)11-5-9-17/h3,6-7H,4-5,8-12H2,1-2H3,(H,18,20)
InChIKey
BCQTVJKBTWGHCX-UHFFFAOYSA-N
Chemical Structure
2D Structure
2D structure of Pilsicainide
CAS: 88069-67-4
CID: 4820
Formula: C17H24N2O
MW: 272.4
Interactive 3D Structure
Loading 3D structure...
View on PubChemRaw 3D data
Computed Properties
PropertyValue
Molecular Weight272.4
XLogP32.7
Hydrogen Bond Donor Count1
Hydrogen Bond Acceptor Count2
Rotatable Bond Count3
Exact Mass272.188863393
Monoisotopic Mass272.188863393
Topological Polar Surface Area32.3 Ų
Heavy Atom Count20
Formal Charge0
Complexity348
Isotope Atom Count0
Defined Atom Stereocenter Count0
Undefined Atom Stereocenter Count0
Defined Bond Stereocenter Count0
Undefined Bond Stereocenter Count0
Covalently-Bonded Unit Count1
Compound Is CanonicalizedYes

Alternative Products

CatalogName
sc-279984Pilsicainide
sc-391025APilsicainide hydrochloride
MBS3611066-01Pilsicainide HCl
HY-101245-01Pilsicainide (hydrochloride)
414954Pilsicainide Free Base
A16362-1000Pilsicainide HCl 1000mg
A16362-500Pilsicainide HCl 500mg
A16362-5Pilsicainide HCl 5mg
A16362-50Pilsicainide HCl 50mg
A16362-25Pilsicainide HCl 25mg

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