PF-4840154

• Target :

  TRP/TRPV Channel

• Related Pathways :

  Membrane transporter/Ion channel

• Purity :

  >99.99%

• Bioactivity :

  PF-4840154 is a potent, selective agonist of the rat and human TrpA1 channel, eliciting TrpA1-mediated nocifensive behavior in mouse, with EC50 values of 97 nM and 23 nM for [rTrpA1] and [hTrpA1], respectively.

• Smiles :

  CC(C)CNc1nc(ncc1C(=O)NCc1ccccc1)N1CCN(CC2CCCOC2)CC1

• Molecular Formula :

  C26H38N6O2

• Molecular Weight :

  466.62

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  1332708-14-1