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DDR1-IN-6

CAT: 0931-T40061-01Size: 2 mgDry Ice: NoHazardous: No
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CAT#:0931-T40061-01Size:2 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2416021-47-9
Target
Others, Discoidin Domain Receptor (DDR)
Related Pathways
Others, Tyrosine Kinase/Adaptors
Bioactivity
DDR1-IN-6 is a potent and selective inhibitor of Discoidin Domain Receptor family member 1 (DDR1), exhibiting remarkable inhibitory activity at an IC50 of 9.72 nM. It effectively suppresses the auto-phosphorylation of DDR1b (Y513) with an IC50 value of 9.7 nM. Furthermore, DDR1-IN-6 displays strong anti-cancer activity.
Smiles
Cc1ccc2c(Nc3cccc(c3)C(F)(F)F)noc2c1C#Cc1cnc2cccnn12
Molecular Formula
C23H14F3N5O
Molecular Weight
433.394
Shipping Conditions
Ice Packs
Storage Temperature
-20°C