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GSK180736A

CAT: 0931-T3513-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T3513-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
817194-38-0
Target
ROCK, GRK, PKA
Related Pathways
GPCR/G Protein, Stem Cells, Cell Cycle/Checkpoint, Cytoskeletal Signaling, Tyrosine Kinase/Adaptors
Purity
0.9898
Bioactivity
GSK180736A is an effective and selective GRK2 inhibitor (IC50: 0.77 μM) and >100-fold selectivity over other GRKs. It is a weak inhibitor of PKA (IC50: 30 μM), but highly effective against ROCK1 (IC50: 100 nM) .
Smiles
CC1=C(C(NC(=O)N1)c1ccc(F)cc1)C(=O)Nc1ccc2[nH]ncc2c1
Molecular Formula
C19H16FN5O2
Molecular Weight
365.36
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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BA4483-5.1GSK180736A
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