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Darexaban

CAT: 0931-T31206-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T31206-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
365462-23-3
Target
Serine Protease, Factor Xa
Related Pathways
Proteases/Proteasome, Metabolism
Purity
0.9881
Bioactivity
Darexaban (Tanexaban, YM-150) is a direct inhibitor of Factor Xa.Darexaban and Darexaban glucuronide selectively and competitively inhibit FXA and inhibit prothrombin activity at the site of blood clot (thrombus) formation. This leads to a reduction in blood clot formation in a dose-dependent manner. Reducing clotting will reduce blockages in blood flow, which may reduce the risk of myocardial infarction, unstable angina, venous thrombosis, and ischemic stroke.
Smiles
COc1ccc(cc1)C(=O)Nc1cccc(O)c1NC(=O)c1ccc(cc1)N1CCCN(C)CC1
Molecular Formula
C27H30N4O4
Molecular Weight
474.55
Shipping Conditions
Ice Packs
Storage Temperature
-20°C