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Pinometostat

CAT: 0931-T3099-01Size: 50 mgDry Ice: NoHazardous: No
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CAT#:0931-T3099-01Size:50 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1380288-87-8
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Purity
0.9986
Bioactivity
Pinometostat (EPZ-5676) is a potent DOT1L histone methyltransferase inhibitor (Ki=80 pM) . Pinometostat has antitumor activity and can be used in experiments to study a variety of leukemia treatments.
Smiles
O[C@H]1[C@H](N2C=3C(N=C2)=C(N)N=CN3)O[C@H](CN(C(C)C)[C@H]4C[C@@H](CCC=5NC=6C(N5)=CC=C(C(C)(C)C)C6)C4)[C@H]1O
Molecular Formula
C30H42N8O3
Molecular Weight
562.71
Shipping Conditions
Ice Packs
Storage Temperature
-20°C