Products for Research Use Only

Cerlapirdine

CAT: 0931-T30798-01Size: 1 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T30798-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
925448-93-7
Target
5-HT Receptor
Related Pathways
GPCR/G Protein, Neuroscience
Purity
0.9877
Bioactivity
Cerlapirdine (PF-05212365) is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.
Smiles
S(=O)(=O)(C=1C=2C(NN1)=CC=C(OCCCN(C)C)C2)C=3C4=C(C=CC3)C=CC=C4
Molecular Formula
C22H23N3O3S
Molecular Weight
409.5
Shipping Conditions
Ice Packs
Storage Temperature
-20°C