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PF-670462

CAT: 0931-T3073-01Size: 2 mgDry Ice: NoHazardous: No
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CAT#:0931-T3073-01Size:2 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
950912-80-8
Target
Casein Kinase
Related Pathways
Metabolism, Stem Cells
Purity
0.9972
Bioactivity
PF-670462 is a potent (IC50 = 7.7 ± 2.2 nM) and selective (>30-fold with respect to 42 additional kinases) inhibitor of CK1ε in isolated enzyme preparations.
Smiles
Cl.Cl.Nc1nccc(n1)-c1c(ncn1C1CCCCC1)-c1ccc(F)cc1
Molecular Formula
C19H22Cl2FN5
Molecular Weight
410.32
Shipping Conditions
Ice Packs
Storage Temperature
-20°C