Droperidol

CAT: 0804-HY-B1240-01Size: 100 mgDry Ice: NoHazardous: No
CAT#:0804-HY-B1240-01Size:100 mg
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Description
Droperidol (Dehydrobenzperidol) is a butyrophenone pamine-2 receptor antagonist that inhibits the activation of GABA (A) and neuronal nicotinic receptors (nAChR), with IC50 values of 12.6 nM and 5.8 μM. Droperidol has anesthetic and sedative properties[1][2].
CAS Number
[548-73-2]
Product Name Alternative
Dehydrobenzperidol
UNSPSC
12352005
Hazard Statement
H302
Target
Dopamine Receptor; GABA Receptor; nAChR
Type
Reference compound
Related Pathways
GPCR/G Protein; Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/Droperidol.html
Concentration
10mM
Purity
99.74
Solubility
DMSO : 33.33 mg/mL (ultrasonic) |H2O : < 0.1 mg/mL
Smiles
O=C1NC2=CC=CC=C2N1C3=CCN(CCCC(C4=CC=C(F)C=C4)=O)CC3
Molecular Formula
C22H22FN3O2
Molecular Weight
379.43
Precautions
H302
References & Citations
[1]Pamela Flood, et al. Droperidol inhibits GABA (A) and neuronal nicotinic receptor activation. Anesthesiology. 2002 Apr;96 (4) :987-93. |[2]J YELNOSKY, et al. A STUDY OF SOME OF THE PHARMACOLOGIC ACTIONS OF DROPERIDOL. Toxicol Appl Pharmacol. 1964 Jan:5:37-47.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, protect from light)
Scientific Category
Reference compound1
Clinical Information
Launched

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