RS-93522

• Target:

  Others|||Calcium Channel

• Related Pathways:

  Membrane transporter/Ion channel|||Others|||Metabolism

• Bioactivity:

  RS-93522 is an antagonist of calcium channel. RS-93522 had the additional property of inhibiting phosphodiesterase activity in myocardial homogenates (IC50 = 1.6 x 10 (-5) M), the potency and efficacy of phosphodiesterase inhibition was similar to that for milrinone in the same system. As expected of Ca channel antagonists, it has a negative inotropic effect on cultured myocardial cells.

• Smiles:

  C(OCCC1=CC=C(OCC(CO)O)C=C1)(=O)C=2C(C(C(OC)=O)=C(C)NC2C)C3=CC(N(=O)=O)=CC=C3

• Molecular Formula:

  C27H30N2O9

• Molecular Weight:

  526.54

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  104060-12-0