Ralaniten

• Target:

  Androgen Receptor

• Related Pathways:

  Endocrinology/Hormones

• Purity:

  0.9996

• Bioactivity:

  Ralaniten (EPI-002) is a potent, specific, and orally active antagonist of the androgen receptor N-terminal structural domain (AR-NTD), inhibiting AR transcriptional activity with an IC50 value of 7.4 ?M. Ralaniten exhibits anticancer activity and is used to study desmoplasia-resistant prostate cancer (CRPC) .

• Smiles:

  CC(C)(c1ccc(OC[C@H](O)CO)cc1)c1ccc(OC[C@H](O)CCl)cc1

• Molecular Formula:

  C21H27ClO5

• Molecular Weight:

  394.89

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1203490-23-6