Ralaniten

• Target :

  Androgen Receptor

• Related Pathways :

  Endocrinology/Hormones

• Purity :

  0.9996

• Bioactivity :

  Ralaniten (EPI-002) is a potent, specific, and orally active antagonist of the androgen receptor N-terminal structural domain (AR-NTD), inhibiting AR transcriptional activity with an IC50 value of 7.4 ?M. Ralaniten exhibits anticancer activity and is used to study desmoplasia-resistant prostate cancer (CRPC) .

• Smiles :

  CC(C)(c1ccc(OC[C@H](O)CO)cc1)c1ccc(OC[C@H](O)CCl)cc1

• Molecular Formula :

  C21H27ClO5

• Molecular Weight :

  394.89

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  1203490-23-6