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Dersimelagon

CAT: 0931-T25310-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T25310-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1835256-48-8
Target
Melanocortin Receptor
Related Pathways
Neuroscience, GPCR/G Protein
Purity
0.9823
Bioactivity
Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values ​​of 8.16, 3.91, 1.14, and 0.251 nM for human (h), cynomolgus monkey (cm), mouse (m), and rat (r) MC1R, respectively. Dersimelagon exhibits good affinity for hMC1R and hMC4R, with Ki values ​​of 2.26 and 32.9 nM, respectively. Dersimelagon can be used in the study of skin pigmentation[1].
Smiles
C(=O)([C@@]1(F)[C@@H](CN(C1)C2CCCC2)C3=CC=C(OC)C=C3)N4C[C@@H]([C@@H](COC)C4)C5=C(C=C(C(F)(F)F)C=C5)N6CCC(C(O)=O)CC6
Molecular Formula
C36H45F4N3O5
Molecular Weight
675.75
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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MBS5775043Dersimelagon
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MBS5812154Dersimelagon phosphate
TRC-D854260-25MGDersimelagon Dihydrochloride

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