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EPZ011989

CAT: 0931-T2435-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T2435-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1598383-40-4
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Purity
0.9981
Bioactivity
EPZ011989 is a effective, specific orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 Y646 and EZH2 wt; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase.
Smiles
CCN([C@H]1CC[C@@H](CC1)N(C)CCOC)c1cc(cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C)C#CCN1CCOCC1
Molecular Formula
C35H51N5O4
Molecular Weight
605.81
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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